Список публикаций Лаборатории синтеза антибиотиков, преодолевающих резистентность (САПР)
I.B. Levshin, A.Y. Simonov, A.A. Panov, N.E. Grammatikova, A.I. Alexandrov, E.S.M.O. Ghazy, V.A. Ivlev, M.O. Agaphonov, A.B. Mantsyzov, V.I. Polshakov, Synthesis and Biological Evaluation of a Series of New Hybrid Amide Derivatives of Triazole and Thiazolidine-2,4-dione, Pharmaceuticals, 2024, 17, 723; https://doi.org/10.3390
/ph17060723A.A. Panov, New Methods of Synthesis of Fused Maleimides, Russian Journal of Organic Chemistry, 2024, 60, 553–567; https://doi.org/10.1134/S1070428024040018
D.V. Andreeva, A.S. Tikhomirov, A.E. Shchekotikhin, Synthesis and antiproliferative activity of thiazole-fused anthraquinones, Organic & Biomolecular Chemistry, 2024, in press; https://doi.org/10.1039/D4OB01284D
V.N. Charushin, E.V. Verbitskiy, O.N. Chupakhin, D.V. Vorobyeva, P.S. Gribanov, S.N. Osipov, A.V. Ivanov, S.V. Martynovskaya, E.F. Sagitova, V.D. Dyachenko, I.V. Dyachenko, S.G. Krivokolysko, V.V. Dotsenko, A.V. Aksenov, D.A. Aksenov, N.A. Aksenov, A.A. Larin, L.L. Fershtat, V.M. Muzalevskiy, V.G. Nenajdenko, A.V. Gulevskaya, A.F. Pozharskii, E.A. Filatova, K.V. Belyaeva, B.A. Trofimov, I.A. Balova, N.A. Danilkina, A.I. Govdi, A.S. Tikhomirov, A.E. Shchekotikhin, M.S. Novikov, N.V. Rostovskii, A.F. Khlebnikov, Yu.N. Klimochkin, M.V. Leonova, I.M. Tkachenko, V.A. Mamedov, V.L. Mamedova, N.A. Zhukova, V.E. Semenov, O.G. Sinyashin, O.V. Borshchev, Yu.N. Luponosov, S.A. Ponomarenko, A.S. Fisyuk, A.S. Kostyuchenko, V.G. Ilkin, T.V. Beryozkina, V.A. Bakulev, A.S. Gazizov, A.A. Zagidullin, A.A. Karasik, M.E. Kukushkin, E.K. Beloglazkina, N.E. Golantsov, A.A. Festa, L.G. Voskresensky, V.S. Moshkin, E.M. Buev, V.Ya. Sosnovskikh, I.A. Mironova, P.S. Postnikov, V.V. Zhdankin, M.S. Yusubov, I.A. Yaremenko, V.A. Vil', I.B. Krylov, A.O. Terent'ev, Yu.G. Gorbunova, A.G. Martynov, A.Yu. Tsivadze, P.A. Stuzhin, S.S. Ivanova, O.I. Koifman, O.N. Burov, M.E. Kletskii, S.V. Kurbatov, O.I. Yarovaya, K.P. Volcho, N.F. Salakhutdinov, M.A. Panova, Ya.V. Burgart, V.I. Saloutin, A.R. Sitdikova, E.S. Shchegravina, A.Yu. Fedorov, The chemistry of heterocycles in the 21st century, Russian Chemical Reviews, 2024, 93 (7), RCR5125; https://doi.org/10.59761/RCR5125
D.V. Andreeva, T.S. Vedekhina, A.S. Gostev, L.G. Dezhenkova, Y.L. Volodina, A.A. Markova, M.T. Nguyen, O.M. Ivanova, V.A. Dolgusheva, A.M. Varizhuk, A.S. Tikhomirov, A.E. Shchekotikhin, Thiadiazole-, selenadiazole- and triazole-fused anthraquinones as G-quadruplex targeting anticancer compounds, European Journal of Medicinal Chemistry, 2024, 268, 116222; https://doi.org/10.1016/j.ejmech.2024.116222
I.A. Volynkina, E.N. Bychkova, A.O. Karakchieva, A.S. Tikhomirov, G.V. Zatonsky, S.E. Solovieva, M.M. Martynov, N.E. Grammatikova, A.G. Tereshchenkov, A. Paleskava, A.L. Konevega, P.V. Sergiev, O.A. Dontsova, I.A. Osterman, A.E. Shchekotikhin, A.N. Tevyashova, Hybrid Molecules of Azithromycin with Chloramphenicol and Metronidazole: Synthesis and Study of Antibacterial Properties, Pharmaceuticals, 2024, 17 (2), 187; https://doi.org/10.3390/ph17020187
V.A.Litvinova, A.S.Tikhomirov, A.E.Shchekotikhin, Methods for functionalization of anthraquinones, Russian Chemical Reviews, 2024, 93, RCR5141, DOI: https://doi.org/10.59761/RCR5141
- A.S. Tikhomirov, Y.B. Sinkevich, L.G. Dezhenkova, D.N. Kaluzhny, N.S. Ilyinsky, V.I. Borshchevskiy, D. Schols, A.E. Shchekotikhin, Synthesis and antitumor activity of cyclopentane-fused anthraquinone derivatives, European Journal of Medicinal Chemistry, 2024, 265, 116103, https://doi.org/10.1016/j.ejmech.2023.116103
M.I. Treshchalin, V.A. Polozkova, E.I. Moiseenko, A.E. Shchekotikhin, S.A. Dovzhenko, M.B. Kobrin, E.R. Pereverzeva, Experimental Evaluation of the Hypersensitivity Reactions of a New Glycopeptide Antibiotic Flavancin in Animal Models, Pharmaceuticals, 2023, 16(11), 1569; https://doi.org/10.3390/ph16111569
V.A. Litvinova, A.S. Gostev, A.S. Tikhomirov, A.E. Shchekotikhin, New heteroarene-fused anthraquinones: Synthesis and PyBOP-mediated amination, Tetrahedron, 2023, 149, 4, 133722, https://doi.org/https://doi.org/10.1016/j.tet.2023.133722
A. Islam, X.C. Chen, C.-W. Weng, C.-Y. Chen, C.-W. Wang, M.-K. Chen, A.S. Tikhomirov, A.E. Shchekotikhin, P.J. Chueh, Water-soluble 4-(dimethylaminomethyl)heliomycin exerts greater antitumor effects than parental heliomycin by targeting the tNOX-SIRT1 axis and apoptosis in oral cancer cells, eLife, 2023, https://doi.org/10.7554/eLife.87873.1
В.А. Литвинова, А.С. Тихомиров, Методы синтеза 1,3-оксазолидин-2-онов, Методы синтеза 1,3-оксазолидин-2-онов, Химия гетероциклических соединений, 2023, 59(11/12), 733-735
K. Shapovalova, G. Zatonsky, N. Grammatikova, I. Osterman, E. Razumova, A. Shchekotikhin, A. Tevyashova, Synthesis of 6”-Modified Kanamycin A Derivatives and Evaluation of Their Antibacterial Properties. Pharmaceutics, 2023, 15, 1177. https://doi.org/10.3390/pharmaceutics15041177
A.A. Panov, Quantum-Chemical Study of Keto-Enol Equilibrium and Global Electrophilicity of Hydroxymaleimide Derivatives. Doklady Physical Chemistry, 2023, 508, 28–32, https://doi.org/10.1134/S001250162360002X
Levshin I.B., Simonov A.Y., Lavrenov S.N., Panov A.A., Grammatikova N.E., Alexandrov A.I., Ghazy E.S.M.O., Savin N.A., Gorelkin P.V., Erofeev A.S., Polshakov V.I. Antifungal Thiazolidines: Synthesis and Biological Evaluation of Mycosidine Congeners. Pharmaceuticals, 2022, 15, 5, 563-586. DOI: 10.3390/ph15050563
Treshchalin M.I., Polozkova V.A., Moiseenko E.I., Treshalina H.M., Shchekotikhin A.E., Pereverzeva E.R. Evaluation of Toxic Properties of New Glycopeptide Flavancin on Rats. Pharmaceuticals, 2022, 15, 661. DOI: 10.3390/ph15060661
- A.N. Tevyashova, S.S. Efimova, A.I. Alexandrov, E.S.M.O. Ghazy, E.N. Bychkova, S.E. Solovieva, G.B. Zatonsky, N.E. Grammatikova, L.G. Dezhenkova, E.R. Pereverzeva, E.B. Isakova, O.S. Ostroumova, O.A. Omelchuk, V.V. Muravieva, M.M. Krotova, T.V. Priputnevich, A.E. Shchekotikhin, Semisynthetic Amides of Polyene Antibiotic Natamycin, ACS Infectious Diseases 2022, 2022, https://doi.org/10.1021/acsinfecdis.2c00237
A. Tevyashova, S. Efimova, A. Alexandrov, O. Omelchuk, E. Ghazy, E. Bychkova, G. Zatonsky, N. Grammatikova, L. Dezhenkova, S. Solovieva, O. Ostroumova, A. Shchekotikhin, Semisynthetic Amides of Amphotericin B and Nystatin A1: A Comparative Study of In Vitro Activity/Toxicity Ratio in Relation to Selectivity to Ergosterol Membranes, Antibiotics 2023, 12(1), 151; https://doi.org/10.3390/antibiotics12010151